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THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors

  1. Author:
    Alexander, Stephen P. H.
    Christopoulos, Arthur
    Davenport, Anthony P.
    Kelly, Eamonn
    Mathie, Alistair
    Peters, John A.
    Veale, Emma L.
    Armstrong, Jane F.
    Faccenda, Elena
    Harding, Simon D.
    Pawson, Adam J.
    Southan, Christopher
    Davies, Jamie A.
    Abbracchio, Maria Pia
    Alexander, Wayne
    Al-hosaini, Khaled
    Baeck, Magnus
    Barnes, Nicholas M.
    Bathgate, Ross
    Beaulieu, Jean-Martin
    Bernstein, Kenneth E.
    Bettler, Bernhard
    Birdsall, Nigel J. M.
    Blaho, Victoria
    Boulay, Francois
    Bousquet, Corinne
    Braeuner-Osborne, Hans
    Burnstock, Geoffrey
    Calo, Girolamo
    Castano, Justo P.
    Catt, KevinJ
    Ceruti, Stefania
    Chazot, Paul
    Chiang, Nan
    Chini, Bice
    Chun, Jerold
    Cianciulli, Antonia
    Civelli, Olivier
    Clapp, Lucie H.
    Couture, Rejean
    Csaba, Zsolt
    Dahlgren, Claes
    Dent, Gordon
    Singh, Khuraijam Dhanachandra
    Douglas, Steven D.
    Dournaud, Pascal
    Eguchi, Satoru
    Escher, Emanuel
    Filardo, Edward J.
    Fong, Tung
    Fumagalli, Marta
    Gainetdinov, Raul R.
    de Gasparo, Marc
    Gerard, Craig
    Gershengorn, Marvin
    Gobeil, Fernand
    Goodfriend, Theodore L.
    Goudet, Cyril
    Gregory, Karen J.
    Gundlach, Andrew L.
    Hamann, Joerg
    Hanson, Julien
    Hauger, Richard L.
    Hay, Debbie L.
    Heinemann, Akos
    Hollenberg, Morley D.
    Holliday, Nicholas D.
    Horiuchi, Mastgugu
    Hoyer, Daniel
    Hunyady, Laszlo
    Husain, Ahsan
    IJzerman, Adriaan P.
    Inagami, Tadashi
    Jacobson, Kenneth A.
    Jensen, Robert T.
    Jockers, Ralf
    Jonnalagadda, Deepa
    Karnik, Sadashiva
    Kaupmann, Klemens
    Kemp, Jacqueline
    Kennedy, Charles
    Kihara, Yasuyuki
    Kitazawa, Takio
    Kozielewicz, Pawel
    Kreienkamp, Hans-Juergen
    Kukkonen, Jyrki P.
    Langenhan, Tobias
    Leach, Katie
    Lecca, Davide
    Lee, John D.
    Leeman, Susan E.
    Leprince, Jerome
    Li, Xaria X.
    Williams, Tom Lloyd
    Lolait, Stephen J.
    Lupp, Amelie
    Macrae, Robyn
    Maguire, Janet
    Mazella, Jean
    McArdle, Craig A.
    Melmed, Shlomo
    Michel, Martin C.
    Miller, Laurence J.
    Mitolo, Vincenzo
    Mouillac, Bernard
    Mueller, Christa E.
    Murphy, Philip
    Nahon, Jean-Louis
    Ngo, Tony
    Norel, Xavier
    Nyimanu, Duuamene
    Ocarroll, Anne-Marie
    Offermanns, Stefan
    Panaro, Maria Antonietta
    Parmentier, Marc
    Pertwee, Roger G.
    Pin, Jean-Philippe
    Prossnitz, Eric R.
    Quinn, Mark
    Ramachandran, Rithwik
    Ray, Manisha
    Reinscheid, Rainer K.
    Rondard, Philippe
    Rovati, G. Enrico
    Ruzza, Chiara
    Sanger, Gareth J.
    Schoeneberg, Torsten
    Schulte, Gunnar
    Schulz, Stefan
    Segaloff, Deborah L.
    Serhan, Charles N.
    Stoddart, Leigh A.
    Sugimoto, Yukihiko
    Summers, Roger
    Tan, Valerie P.
    Thal, David
    Thomas, Walter (Wally)
    Timmermans, PieterB M. W. M.
    Tirupula, Kalyan
    Tulipano, Giovanni
    Unal, Hamiyet
    Unger, Thomas
    Valant, Celine
    Vanderheyden, Patrick
    Vaudry, David
    Vaudry, Hubert
    Vilardaga, Jean-Pierre
    Walker, Christopher S.
    Wang,Jiming
    Ward, Donald T.
    Wester, Hans-Juergen
    Willars, Gary B.
    Woodruff, Trent M.
    Yao, Chengcan
    Ye, Richard D.

  2. Author Address

    Univ Nottingham Med Sch, Sch Life Sci, Nottingham NG7 2UH, England.Monash Univ, Monash Inst Pharmaceut Sci, Parkville, Vic 3052, Australia.Monash Univ, Dept Pharmacol, Parkville, Vic 3052, Australia.Univ Cambridge, Clin Pharmacol Unit, Cambridge CB2 0QQ, England.Univ Bristol, Sch Physiol Pharmacol & Neurosci, Bristol BS8 1TD, Avon, England.Univ Suffolk, Sch Engn Arts Sci & Technol, Ipswich IP4 1QJ, Suffolk, England.Univ Dundee, Ninewells Hosp & Med Sch, Med Educ Inst, Neurosci Div, Dundee DD1 9SY, Scotland.Univ Greenwich & Kent Medway, Medway Sch Pharm, Anson Bldg,Cent Ave, Chatham ME4 4TB, Kent, England.Univ Edinburgh, Ctr Discovery Brain Sci, Edinburgh EH8 9XD, Midlothian, Scotland.Univ Milan, Milan, Italy.Emory Univ, Atlanta, GA 30322 USA.King Saud Univ, Riyadh, Saudi Arabia.Karolinska Univ Hosp, Stockholm, Sweden.Univ Birmingham, Birmingham, W Midlands, England.Florey Inst Neurosci & Mental Hlth, Melbourne, Vic, Australia.Univ Toronto, Toronto, ON, Canada.Cedars Sinai Med Ctr, Los Angeles, CA 90048 USA.Univ Basel, Basel, Switzerland.Francis Crick Inst, London, England.Sanford Burnham Prebys Med Discovery Inst, La Jolla, CA USA.Univ Grenoble Alpes, Grenoble, France.French Inst Hlth & Med Res INSERM, Toulouse, France.Univ Copenhagen, Copenhagen, Denmark.Univ Coll London, Melbourne, Vic, Australia.Univ Padua, Padua, Italy.Univ Cordoba, Cordoba, Spain.NIH, Bldg 10, Bethesda, MD 20892 USA.Univ Durham, Durham, England.Harvard Univ, Boston, MA 02115 USA.Univ Milano Bicocca, Vedano Al Lambro, Italy.Univ Calif San Diego, La Jolla, CA 92093 USA.Univ Bari, Bari, Italy.Univ Calif Irvine, Irvine, CA USA.UCL, London, England.Univ Montreal, Montreal, PQ, Canada.French Inst Hlth & Med Res INSERM, Paris, France.Univ Gothenburg, Gothenburg, Sweden.Keele Univ, Keele, Staffs, England.Cleveland Clin, Lerner Res Inst, Cleveland, OH 44106 USA.Univ Penn, Philadelphia, PA 19104 USA.Temple Univ, Philadelphia, PA USA.Univ Sherbrooke, Sherbrooke, PQ, Canada.Univ Iowa, Iowa City, IA USA.Labcorp Drug Dev, Somerset, NJ USA.St Petersburg State Univ, St Petersburg, Russia.MG Consulting Co, Basel, Switzerland.Univ Wisconsin, Madison, WI USA.French Natl Ctr Sci Res, Montpellier, France.Monash Univ, Parkville, Vic, Australia.Univ Amsterdam, Amsterdam, Netherlands.Univ Liege, Liege, Belgium.Univ Otago, Dunedin, New Zealand.Med Univ Graz, Graz, Austria.Univ Calgary, Calgary, AB, Canada.Univ Nottingham, Nottingham, England.Ehime Univ, Matsuyama, Ehime, Japan.Univ Melbourne, Melbourne, Vic, Australia.Semmelweis Univ, Budapest, Hungary.Emory Univ, Birmingham, AL USA.Leiden Univ, Leiden, Netherlands.Vanderbilt Univ, 221 Kirkland Hall, Nashville, TN 37235 USA.Lerner Res Inst, Cleveland, OH USA.Novartis, Basel, Switzerland.Strathclyde Univ, Glasgow, Lanark, Scotland.Rakuno Gakuen Univ, Ebetsu, Hokkaido, Japan.Karolinska Inst, Stockholm, Sweden.Univ Hamburg, Hamburg, Germany.Univ Helsinki, Helsinki, Finland.Univ Leipzig, Leipzig, Germany.Univ Queensland, Brisbane, Qld, Australia.Boston Univ, Boston, MA 02215 USA.Univ Rouen, Rouen, France.Univ Cambridge, Cambridge, England.Univ Bristol, Bristol, Avon, England.Friedrich Schiller Univ Jena, Jena, Germany.French Natl Ctr Sci Res CNRS, Valbonne, France.Johannes Gutenberg Univ Mainz, Mainz, Germany.Mayo Fdn Med Educ & Res, Scottsdale, AZ USA.Univ Bonn, Bonn, Germany.Edge Hill Univ, Bethesda, MD USA.Max Planck Inst Heart & Lung Res, Bad Nauheim, Germany.Free Univ Brussels, Brussels, Belgium.Univ Aberdeen, Aberdeen, Scotland.Univ Montpellier, Montpellier, France.Univ New Mexico, Albuquerque, NM 87131 USA.Montana State Univ, Bozeman, MT 59717 USA.Univ Calgary, London, ON, Canada.Univ Ferrara, Ferrara, Italy.Queen Mary Univ London, London, England.Univ Leipzig, Leipzig, Germany.Kumamoto Univ, Kumamoto, Japan.Monash Univ, Melbourne, Vic, Australia.Kosan Biosci Inc, San Francisco, CA USA.Univ Brescia, Brescia, Italy.Cleveland Clin, Cleveland, OH 44106 USA.Maastricht Univ, Maastricht, Netherlands.Univ Pittsburgh, Pittsburgh, PA USA.Univ Auckland, Auckland, New Zealand.NIH, Frederick, MD USA.Univ Manchester, Manchester, Lancs, England.Tech Univ Munich, Munich, Germany.Univ Leicester, Leicester, Leics, England.Univ Edinburgh, Edinburgh, Midlothian, Scotland.Univ Illinois, Chicago, IL USA.
    1. Year: 2021
    2. Date: Oct
  2. Journal: British journal of pharmacology
  3. WILEY,
    1. 178 Suppl 1
    2. 1
    3. Pages: S27-S156
  5. Type of Article: Article
  6. ISSN: 0007-1188
  1. Abstract:

    The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at . G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.

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External Sources

  1. View Full Text
  2. DOI: 10.1111/bph.15538
  3. PMID: 34529832
  4. View record in Web of Science®
  5. WOS: 000696321000003

Library Notes

  1. Fiscal Year: FY2021-2022
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