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  1. 1.   Comparative Analyses of Antiviral Potencies of Second-Generation Integrase Strand Transfer Inhibitors (INSTIs) and the Developmental Compound 4d Against a Panel of Integrase Quadruple Mutants
  2. Smith,Steven; Zhao,Xuezhi; Hughes,Stephen; Burke,Terrence
  3. Viruses. 2025, Jan 16; 17(1):
  1. 2.   Dihydroxyphenyl- and Heteroaromatic-Based Thienopyrimidinones to Tackle HIV-1 LEDGF/p75-Dependent IN Activity
  2. Tocco, Graziella; Canton, Serena; Laus, Antonio; Caboni, Pierluigi; Le Grice, Stuart F J; Tramontano, Enzo; Esposito, Francesca
  3. Molecules (Basel, Switzerland). 2023, Sep 19; 28(18):
  1. 3.   A Practical Approach to Bicyclic Carbamoyl Pyridones with Application to the Synthesis of HIV-1 Integrase Strand Transfer Inhibitors
  2. Mahajan,Pankaj; Smith,Steven; Hughes,Stephen; Zhao,Xue Zhi; Burke,Terrence
  3. Molecules (Basel, Switzerland). 2023, Feb 02; 28(3):
  1. 4.   The C-Terminal Domain of RNase H and the C-Terminus Amino Acid Residue Regulate Virus Release and Autoprocessing of a Defective HIV-1 Possessing M50I and V151I Changes in Integrase
  2. Imamichi,Tomozumi; Chen,Qian; Hao, Ming; Chang,Weizhong; Yang,Jun
  3. Viruses. 2022, Nov 30; 14(12):
  1. 5.   Scaffolding viral protein NC nucleates phase separation of the HIV-1 biomolecular condensate
  2. Monette, Anne; Niu, Meijuan; Nijhoff Asser, Maya; Gorelick,Robert; Mouland, Andrew J
  3. Cell Reports. 2022, Aug 23; 40(8): 111251.
  1. 6.   Natural Occurring Polymorphisms in HIV-1 Integrase and RNase H Regulate Viral Release and Autoprocessing
  2. Imamichi, Tomozumi; Bernbaum, John G.; Laverdure, Sylvain; Yang, Jun; Chen, Qian; Highbarger, Helene; Hao, Ming; Sui, Hongyan; Dewar, Robin; Chang, Weizhong; Lane, H. Clifford
  3. Journal of Virology . 2021, Dec; 95(23):
  1. 7.   A Combination of M50I and V151I Polymorphic Mutations in HIV-1 Subtype B Integrase Results in Defects in Autoprocessing
  2. Yang, Jun; Hao,Ming; Khan, Muhammad A; Rehman,Tauseef; Highbarger,Helene; Chen,Qian; Goswami,Suranjana; Sherman,Brad; Rehm, Catherine A; Dewar,Robin; Chang,Weizhong; Imamichi, Tomozumi
  3. Viruses. 2021, Nov 22; 13(11):
  1. 8.   HIV-1 Integrase Inhibitors with Modifications That Affect Their Potencies against Drug Resistant Integrase Mutants
  2. Smith,Steven; Zhao,Xue Zhi; Passos, Dario Oliveira; Pye, Valerie E.; Cherepanov, Peter; Lyumkis, Dmitry; Burke,Terrence; Hughes,Stephen
  3. ACS Infectious Diseases. 2021, Jun 11; 7(6): 1469-1482.
  1. 9.   Scaffold hopping and optimisation of 3',4'-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H
  2. Tocco, Graziella; Esposito, Francesca; Caboni, Pierluigi; Laus, Antonio; Beutler,John; Wilson,Jennifer; Corona, Angela; Le Grice,Stuart; Tramontano, Enzo
  3. Journal of enzyme inhibition and medicinal chemistry. 2020, Dec; 35(1): 1953-1963.
  1. 10.   How to package the RNA of HIV-1
  2. Kleinpeter,Alex; Freed,Eric
  3. eLife. 2020, Nov 17; 9: pii: e63585.
  1. 11.   HIV-1 Integrase Inhibitors that are active against Drug-Resistant Integrase Mutants
  2. Smith,Steven; Zhao,Xue Zhi; Passos, Dario Oliveira; Lyumkis, Dmitry; Burke,Terrence; Hughes,Stephen
  3. Antimicrobial agents and chemotherapy. 2020, SEP; 64(9):
  1. 12.   (Q)SAR Models of HIV-1 Protein Inhibition by Drug-Like Compounds
  2. Stolbov, Leonid A; Druzhilovskiy, Dmitry S; Filimonov, Dmitry A; Nicklaus,Marc; Poroikov, Vladimir V
  3. Molecules (Basel, Switzerland). 2020, Jan 1; 25(1):
  1. 13.   Capsid-CPSF6 Interaction Licenses Nuclear HIV-1 Trafficking to Sites of Viral DNA Integration
  2. Achuthan, Vasudevan; Perreira, Jill M; Sowd, Gregory A; Puray-Chavez, Maritza; McDougall, William M; Paulucci-Holthauzen, Adriana; Wu, Xiaolin; Fadel, Hind J; Poeschla, Eric M; Multani, Asha S; Hughes, Stephen; Sarafianos, Stefan G; Brass, Abraham L; Engelman, Alan N
  3. Cell host & microbe. 2018, Sep 12; 24(3): 392-404.e8.
  1. 14.   HIV-1 Integrase-Targeted Short Peptides Derived from a Viral Protein R Sequence
  2. Zhao, Xue Zhi; Métifiot, Mathieu; Kiselev, Evgeny; Kessl, Jacques J; Maddali, Kasthuraiah; Marchand, Christophe; Kvaratskhelia, Mamuka; Pommier, Yves; Burke, Terrence
  3. Molecules . 2018, Aug; 23(8): pii: E1858.
  1. 15.   Efficacies of Cabotegravir and Bictegravir against drug-resistant HIV-1 integrase mutants
  2. Smith, Steven; Zhao, Xue Zhi; Burke, Terrence; Hughes, Stephen
  3. Retrovirology. 2018, May 16; 15(1): 37.
  1. 16.   Localization of ASV Integrase-DNA Contacts by Site-Directed Crosslinking and their Structural Analysis
  2. Peletskaya, E.; Andrake, M.; Gustchina, A.; Merkel, G.; Alexandratos, J.; Zhou, D. W.; Bojja, R. S.; Satoh, T.; Potapov, M.; Kogon, A.; Potapov, V.; Wlodawer, A.; Skalka, A. M.
  3. Plos One. 2011, Dec; 6(12):
  1. 17.   Impact of treatment with raltegravir during primary or chronic HIV infection on RNA decay characteristics and the HIV viral reservoir
  2. Koelsch, K. K.; Boesecke, C.; McBride, K.; Gelgor, L.; Fahey, P.; Natarajan, V.; Baker, D.; Bloch, M.; Murray, J. M.; Zaunders, J.; Emery, S.; Cooper, D. A.; Kelleher, A. D.; Team, P. S.
  3. Aids. 2011, Nov; 25(17): 2069-2078.
  1. 18.   Structural and Functional Analyses of the Second-Generation Integrase Strand Transfer Inhibitor Dolutegravir (S/GSK1349572)
  2. Hare, S.; Smith, S. J.; Metifiot, M.; Jaxa-Chamiec, A.; Pommier, Y.; Hughes, S. H.; Cherepanov, P.
  3. Molecular Pharmacology. 2011, Oct; 80(4): 565-572.
  1. 19.   Association of polymorphisms in the LEDGF/p75 gene (PSIP1) with susceptibility to HIV-1 infection and disease progression
  2. Madlala, P.; Gijsbers, R.; Christ, F.; Hombrouck, A.; Werner, L.; Mlisana, K.; An, P.; Karim, S. S. A.; Winkler, C. A.; Debyser, Z.; Ndung'u, T.
  3. Aids. 2011, Sep; 25(14): 1711-1719.
  1. 20.   Software and resources for computational medicinal chemistry
  2. Liao, C. Z.; Sitzmann, M.; Pugliese, A.; Nicklaus, M. C.
  3. Future Medicinal Chemistry. 2011, Jun; 3(8): 1057-1085.
  1. 21.   Development of tricyclic hydroxy-1H-pyrrolopyridine-trione containing HIV-1 integrase inhibitors
  2. Zhao, X. Z.; Maddali, K.; Metifiot, M.; Smith, S. J.; Vu, B. C.; March, C.; Hughes, S. H.; Pommier, Y.; Burke, T. R.
  3. Bioorganic & Medicinal Chemistry Letters. 2011, May; 21(10): 2986-2990.
  1. 22.   Transmitted raltegravir resistance in an HIV-1 CRF_AG-infected patient
  2. Boyd, S. D.; Maldarelli, F.; Sereti, I.; Ouedraogo, G. L.; Rehm, C. A.; Boltz, V.; Shoemaker, D.; Pau, A. K.
  3. Antiviral Therapy. 2011 16(2): 257-261.
  1. 23.   Tautomerism and Magnesium Chelation of HIV-1 Integrase Inhibitors: A Theoretical Study
  2. Liao, C. Z.; Nicklaus, M. C.
  3. Chemmedchem. 2010, Jul 5; 5(7): 1053-1066.
  1. 24.   Computer tools in the discovery of HIV-1 integrase inhibitors
  2. Liao, C. Z.; Nicklaus, M. C.
  3. Future Medicinal Chemistry. 2010, Jul; 2(7): 1123-1140.
  1. 25.   Authentic HIV-1 integrase inhibitors
  2. Liao, C. Z.; March, C.; Burke, T. R.; Pommier, Y.; Nicklaus, M. C.
  3. Future Medicinal Chemistry. 2010, Jul; 2(7): 1107-1122.
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