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  1. 1.   Evaluation of the Therapeutic Potential of Sulfonyl Urea Derivatives as Soluble Epoxide Hydrolase (sEH) Inhibitors
  2. Kundu, Biswajit; Dvorácskó, Szabolcs; Basu, Abhishek; Pommerolle, Lenny; Kim, Kyu Ah; Wood, Casey M; Gibbs, Eve; Behee, Madeline; Tarasova,Nadya; Cinar, Resat; Iyer, Malliga R
  3. Molecules (Basel, Switzerland). 2024, Jun 26; 29(13):
  1. 2.   An Investigation of Structure-Activity Relationships and Cell Death Mechanisms of the Marine Alkaloids Discorhabdins in Merkel Cell Carcinoma Cells
  2. Orfanoudaki,Maria; Smith,Emily; Hill, Natasha T; Garman, Khalid A; Brownell, Isaac; Copp, Brent R; Grkovic,Tanja; Henrich,Curtis
  3. Marine Drugs. 2023, Aug 29; 21(9):
  1. 3.   µ-Conotoxins Targeting the Human Voltage-Gated Sodium Channel Subtype NaV1.7
  2. McMahon, Kirsten L; Tran, Hue N T; Deuis, Jennifer R; Craik, David J; Vetter, Irina; Schroeder, Christina I
  3. Toxins. 2022, Aug 30; 14(9):
  1. 4.   Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents
  2. Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel,Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
  3. Pharmaceutics. 2022, Jun 02; 14(6):
  1. 5.   Novel pyrazolo[4,3-d]pyrimidine microtubule targeting agents (MTAs): Synthesis, structure-activity relationship, in vitro and in vivo evaluation as antitumor agents
  2. Islam, Farhana; Quadery, Tasdique M.; Bai,Ruoli; Luckett-Chastain, Lerin R.; Hamel,Ernest; Ihnat, Michael A.; Gangjee, Aleem
  3. Bioorganic & Medicinal Chemistry Letters. 2021, Jun 1; 41
  1. 6.   Optimization of ether and aniline based inhibitors of lactate dehydrogenase
  2. Christov, Plamen P.; Kim, Kwangho; Jana, Somnath; Romaine, Ian M.; Rai, Ganesha; Mott, Bryan T.; Allweil, Alexander A.; Lamers, Alexander; Brimacombe, Kyle R.; Urban, Daniel J.; Lee, Tobie D.; Hu, Xin; Lukacs, Christine M.; Davies, Douglas R.; Jadhav, Ajit; Hall, Matthew D.; Green, Neal; Moore,Bill; Stott,Gordon; Flint,Andrew; Maloney, David J.; Sulikowski, Gary A.; Waterson, Alex G.
  3. Bioorganic & Medicinal Chemistry Letters. 2021, Jun 1; 41: 127974.
  1. 7.   A facile synthesis of diaryl pyrroles led to the discovery of potent colchicine site antimitotic agents
  2. Romagnoli, Romeo; Oliva, Paola; Salvador, Maria Kimatrai; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel,Ernest; Ronca, Roberto; Maccarinelli, Federica; Rruga, Fatlum; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
  3. European Journal of Medicinal Chemistry. 2021, Mar 15; 214
  1. 8.   Structure-Activity Relationships of Pyrazolo[1,5-a]pyrimidin-7(4H)-ones as Antitubercular Agents
  2. Oh, Sangmi; Libardo, M. Daben J.; Azeeza, Shaik; Pauly,Gary; Roma, Jose Santinni O.; Sajid, Andaleeb; Tateishi, Yoshitaka; Duncombe, Caroline; Goodwin, Michael; Ioerger, Thomas R.; Wyatt, Paul G.; Ray, Peter C.; Gray, David W.; Boshoff, Helena I. M.; Barry, Clifton E.
  3. ACS Infectious Diseases. 2021, Feb 12; 7(2): 479-492.
  1. 9.   The 3-D conformational shape of N-naphthyl-cyclopenta[d]pyrimidines affects their potency as microtubule targeting agents and their antitumor activity
  2. Xiang, Weiguo; Quadery, Tasdique M; Hamel,Ernest; Luckett-Chastain, Lerin R; Ihnat, Michael A; Mooberry, Susan L; Gangjee, Aleem
  3. Bioorganic & medicinal chemistry. 2021, Jan 1; 29: 115887.
  1. 10.   Antiangiogenic Activity and in Silico Cereblon Binding Analysis of Novel Thalidomide Analogs
  2. Peach,Megan; Beedie, Shaunna L; Chau, Cindy H; Collins, Matthew K; Markolovic, Suzana; Luo, Weiming; Tweedie, David; Steinebach, Christian; Greig, Nigel H; Gütschow, Michael; Vargesson, Neil; Nicklaus,Marc; Figg, William D
  3. Molecules (Basel, Switzerland). 2020, DEC; 25(23): 5683.
  1. 11.   Synthesis and Biological Evaluation of 2-Substituted Benzyl-/Phenylethylamino-4-amino-5-aroylthiazoles as Apoptosis-Inducing Anticancer Agents
  2. Oliva, Paola; Onnis, Valentina; Balboni, Elisa; Hamel,Ernest; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Romagnoli, Romeo
  3. Molecules (Basel, Switzerland). 2020, May 06; 25(9):
  1. 12.   Synthesis and Biological Evaluation of New Antitubulin Agents Containing 2-(3',4',5'-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold
  2. Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel,Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto
  3. Molecules (Basel, Switzerland). 2020, Apr 07; 25(7): pii : molecules25071690.
  1. 13.   Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization
  2. Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Kimatrai Salvador, Maria; Brancale, Andrea; Ferla, Salvatore; Hamel,Ernest; Viola, Giampietro; Bortolozzi, Roberta; Persoons, Leentje; Balzarini, Jan; Liekens, Sandra; Schols, Dominique
  3. Bioorganic chemistry. 2020, APR; 97: 103665.
  1. 14.   Design, synthesis and biological evaluation of novel vicinal diaryl-substituted 1H-Pyrazole analogues of combretastatin A-4 as highly potent tubulin polymerization inhibitors
  2. Romagnoli, Romeo; Oliva, Paola; Salvador, Maria Kimatrai; Camacho, Maria Encarnacion; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel,Ernest; Ronca, Roberto; Grillo, Elisabetta; Bortolozzi, Roberta; Rruga, Fatlum; Mariotto, Elena; Viola, Giampietro
  3. European journal of medicinal chemistry. 2019, NOV 1; 181: 111577.
  1. 15.   Evaluating the effects of fluorine on biological properties and metabolic stability of some antitubulin 3-substituted 7-phenyl-pyrroloquinolinones
  2. Bortolozzi, Roberta; Carta, Davide; Prà, Matteo Dal; Antoniazzi, Giuseppe; Mattiuzzo, Elena; Sturlese, Mattia; Di Paolo, Veronica; Calderan, Laura; Moro, Stefano; Hamel,Ernest; Quintieri, Luigi; Ronca, Roberto; Viola, Giampietro; Ferlin, Maria Grazia
  3. European journal of medicinal chemistry. 2019, Sep 15; 178: 297-314.
  1. 16.   Genotoxicity of amorphous silica nanoparticles: Status and prospects
  2. Yazdimamaghani, Mostafa; Moos, Philip J.; Dobrovolskaia, Marina; Ghandehari, Hamidreza
  3. Nanomedicine : nanotechnology, biology, and medicine. 2019, Feb; 16: 106-125.
  1. 17.   Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach
  2. Preti, Delia; Romagnoli, Romeo; Rondanin, Riccardo; Cacciari, Barbara; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Schols, Dominique; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco
  3. Journal of enzyme inhibition and medicinal chemistry. 2018, Dec; 33(1): 1225-1238.
  1. 18.   3-Aryl/Heteroaryl-5-amino-1-(3',4',5'-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
  2. Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
  3. Bioorganic chemistry. 2018, Oct; 80: 361-374.
  1. 19.   Design, synthesis and preclinical evaluation of 5-methyl-N4-aryl-furo[2,3-d]pyrimidines as single agents with combination chemotherapy potential
  2. Devambatla, Ravi Kumar Vyas; Choudhary, Shruti; Ihnat, Michael; Hamel, Ernest; Mooberry, Susan L; Gangjee, Aleem
  3. Bioorganic & Medicinal Chemistry Letters. 2018, Oct 1; 28(18): 3085-3093.
  1. 20.   Targeting tubulin polymerization by novel 7-aryl-pyrroloquinolinones: Synthesis, biological activity and SARs
  2. Bortolozzi, Roberta; Mattiuzzo, Elena; Dal Pra, Matteo; Sturlese, Mattia; Moro, Stefano; Hamel, Ernest; Carta, Davide; Viola, Giampietro; Ferlin, Maria Grazia
  3. European journal of medicinal chemistry. 2018, Jan 1; 143: 244-258.
  1. 21.   2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition
  2. Romagnoli, Romeo; Kimatrai Salvador, Maria; Schiaffino Ortega, Santiago; Baraldi, Pier Giovanni; Oliva, Paola; Baraldi, Stefania; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro
  3. European Journal of Medicinal Chemistry. 2018, Jan 1; 143: 683-698.
  1. 22.   Targeting tubulin polymerization by novel 7-aryl-pyrroloquinolinones: Synthesis, biological activity and SARs
  2. Bortolozzi, Roberta; Mattiuzzo, Elena; Dal Pra, Matteo; Sturlese, Mattia; Moro, Stefano; Hamel, Ernest; Carta, Davide; Viola, Giampietro; Ferlin, Maria Grazia
  3. European Journal of Medicinal Chemistry. 2018, Jan 01; 143: 244-258.
  1. 23.   Synthesis, structure-activity relationships and biological evaluation of 7-phenyl-pyrroloquinolinone 3-amide derivatives as potent antimitotic agents
  2. Carta, D.; Bortolozzi, R.; Sturlese, M.; Salmaso, V.; Hamel, Ernest; Basso, G.; Calderan, L.; Quintieri, L.; Moro, S.; Viola, G.; Ferlin, M. G.
  3. European Journal of Medicinal Chemistry. 2017, Feb 15; 127: 643-660.
  1. 24.   Oxime Ether Lipids as Transfection Agents: Assembly and Complexation with siRNA.
  2. Puri, Anu; Zampino, Serena; Viard, Mathias; Shapiro, Bruce
  3. Methods in molecular biology (Clifton, N.J.). 2017 1632: 241-253.
  1. 25.   Design, synthesis, and biological evaluation of water-soluble amino acid prodrug conjugates derived from combretastatin, dihydronaphthalene, and benzosuberene-based parent vascular disrupting agents
  2. Devkota, L.; Lin, C. M.; Strecker, T. E.; Wang, Y.; Tidmore, J. K.; Chen, Z.; Guddneppanavar, R.; Jelinek, C. J.; Lopez, R.; Liu, L.; Hamel, E.; Mason, R. P.; Chaplin, D. J.; Trawick, M. L.; Pinney, K. G.
  3. Bioorganic & Medicinal Chemistry. 2016, 1-Mar; 24(5): 938-56.
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